Chemicals and Drugs

Proteinase-Activated Receptors

A class of receptors that are activated by the action of PROTEINASES. The most notable examples are the THROMBIN RECEPTORS. The receptors contain cryptic ligands that are exposed upon the selective proteolysis of specific N-terminal cleavage sites.

National Library of MedicineMedical Subject Headings2026

Structured Summary

Abstract

A class of receptors that are activated by the action of PROTEINASES. The most notable examples are the THROMBIN RECEPTORS. The receptors contain cryptic ligands that are exposed upon the selective proteolysis of specific N-terminal cleavage sites.

MeSH Record

Classification

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MeSH Record

Synonyms

18 entry terms
  • Endopeptidase-Activated Receptor
  • Endopeptidase-Activated Receptors
  • Protease-Activated Receptor
  • Protease-Activated Receptors
  • Proteinase-Activated Receptor
  • Receptors, Proteinase-Activated
  • Endopeptidase Activated Receptor
  • Endopeptidase Activated Receptors
  • Protease Activated Receptor
  • Protease Activated Receptors
  • Proteinase Activated Receptor
  • Proteinase Activated Receptors
  • Receptor, Endopeptidase-Activated
  • Receptor, Protease-Activated
  • Receptor, Proteinase-Activated
  • Receptors, Endopeptidase-Activated
  • Receptors, Protease-Activated
  • Receptors, Proteinase Activated

MeSH Record

Aspects Covered

19 allowable subheadings

Indexed with the subheadings administration & dosage, agonists, analysis, antagonists & inhibitors, biosynthesis, blood, chemistry, classification, deficiency, drug effects, genetics, history, immunology, isolation & purification, metabolism, physiology, radiation effects, therapeutic use, ultrastructure.

MeSH Record

History Note

2004

MeSH Record

Previous Indexing

  • Receptors, Thrombin (1994-2003)

MeSH Hierarchy

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AMA Style

References

  1. National Library of Medicine. Proteinase-Activated Receptors. Medical Subject Headings (MeSH). 2026. Unique ID D044462. http://id.nlm.nih.gov/mesh/2026/D044462
  2. Proteinase-Activated Receptors. In: Wikipedia. https://en.wikipedia.org/wiki/Protease-activated_receptor
  3. Proteinase-Activated Receptors. In: Wikidata. https://www.wikidata.org/wiki/Q24777577